2. GPCR/G Protein
  3. GnRH Receptor
  4. Linzagolix choline

Linzagolix choline  (Synonyms: KLH-2109 choline; OBE-2109 choline)

Cat. No.: HY-120767
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Linzagolix choline (KLH-2109 choline) is a non-peptide gonadotropin-releasing hormone (GnRH) antagonist with oral activity. Linzagolix choline inhibits the release of endogenous gonadotropins such as luteinizing hormone LH and follicle-stimulating hormone FSH by binding to the GnRH receptor within the pituitary gland. This inhibition results in a reduction in the production of sex hormones such as estrogen and progesterone, which in turn affects the course of sex hormone-dependent diseases. Linzagolix choline can be used in the study of sex hormone-dependent diseases such as endometriosis and uterine fibroids.

For research use only. We do not sell to patients.

Linzagolix choline Chemical Structure

Linzagolix choline Chemical Structure

CAS No. : 1321816-57-2

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Linzagolix choline Related Antibodies

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Description

Linzagolix choline (KLH-2109 choline) is a non-peptide gonadotropin-releasing hormone (GnRH) antagonist with oral activity. Linzagolix choline inhibits the release of endogenous gonadotropins such as luteinizing hormone LH and follicle-stimulating hormone FSH by binding to the GnRH receptor within the pituitary gland. This inhibition results in a reduction in the production of sex hormones such as estrogen and progesterone, which in turn affects the course of sex hormone-dependent diseases. Linzagolix choline can be used in the study of sex hormone-dependent diseases such as endometriosis and uterine fibroids[1].

Molecular Weight

611.59

Formula

C27H28F3N3O8S
CAS No.
SMILES

OCC[N+](C)(C)C.O=C([O-])C1=C(C(NC2=O)=CS1)C(N2C3=CC(OCC4=C(C=CC(F)=C4F)OC)=C(C=C3F)OC)=O
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Room temperature in continental US; may vary elsewhere.
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Please store the product under the recommended conditions in the Certificate of Analysis.
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Linzagolix choline Related Classifications

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Help & FAQs
  • Do most proteins show cross-species activity?

    Species cross-reactivity must be investigated individually for each product. Many human cytokines will produce a nice response in mouse cell lines, and many mouse proteins will show activity on human cells. Other proteins may have a lower specific activity when used in the opposite species.

Keywords:

Linzagolix1321816-57-2KLH-2109OBE-2109KLH2109KLH 2109OBE2109OBE 2109GnRH ReceptorGonadotropin releasing hormone receptorGNRHREndogenous gonadotropinantagonistsex hormone dependent diseaseoral activityGnRHInhibitorinhibitorinhibit

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