1. PROTAC
  2. PROTACs
  3. cBu-Cit-PROTAC BRD4 Degrader-5

cBu-Cit-PROTAC BRD4 Degrader-5 is a cBu-Cit conjugated PROTAC degrader. cBu-Cit-PROTAC BRD4 Degrader-5 can potently degrade BRD4 in HER2 positive and negative breast cancer cell lines.

For research use only. We do not sell to patients.

cBu-Cit-PROTAC BRD4 Degrader-5 Chemical Structure

cBu-Cit-PROTAC BRD4 Degrader-5 Chemical Structure

CAS No. : 2417369-73-2

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Description

cBu-Cit-PROTAC BRD4 Degrader-5 is a cBu-Cit conjugated PROTAC degrader. cBu-Cit-PROTAC BRD4 Degrader-5 can potently degrade BRD4 in HER2 positive and negative breast cancer cell lines[1].

Molecular Weight

1628.31

Formula

C79H99ClN16O16S2

CAS No.
SMILES

CC1=C(C)SC2=C1C(C3=CC=C(C=C3)Cl)=N[C@@H](CC(NCCOCCOCCOCC(N[C@@H](C(C)(C)C)C(N4[C@@H](C[C@H](C4)OCNC(OCC5=CC=C(C=C5)NC([C@H](CCCNC(N)=O)NC(C6(CCC6)C(NCCCCCN7C(C=CC7=O)=O)=O)=O)=O)=O)C(NCC8=CC=C(C9=C(N=CS9)C)C=C8)=O)=O)=O)=O)C%10=NN=C(C)N2%10

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Room temperature in continental US; may vary elsewhere.

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Please store the product under the recommended conditions in the Certificate of Analysis.

Purity & Documentation
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cBu-Cit-PROTAC BRD4 Degrader-5 Related Classifications

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Help & FAQs
  • Do most proteins show cross-species activity?

    Species cross-reactivity must be investigated individually for each product. Many human cytokines will produce a nice response in mouse cell lines, and many mouse proteins will show activity on human cells. Other proteins may have a lower specific activity when used in the opposite species.

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Product Name:
cBu-Cit-PROTAC BRD4 Degrader-5
Cat. No.:
HY-160694
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