Calcium Channel antagonist 2

Cat. No.: HY-156663 Purity: ≥98.0%: FAQs
Data Sheet SDS COA Handling Instructions

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Calcium Channel antagonist 2 (Compound 154) is a calcium channel antagonist (IC₅₀=5-20 μM). Calcium Channel antagonist 2 can be used in study of calcium channel-mediated diseases such as pain and diabetes.

For research use only. We do not sell to patients.

Calcium Channel antagonist 2 Chemical Structure

CAS No. : 874370-15-7

Size	Price	Stock	Quantity
10 mg	USD 50	In-stock	Estimated Time of Arrival: December 31
50 mg		Get quote
100 mg		Get quote

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Purity & Documentation
References
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Description

Molecular Weight

444.52

Formula

C₂₃H₂₅FN₂O₄S

CAS No.

874370-15-7

Appearance

Solid

Color

White to off-white

SMILES

O=C(C1=C(C)C2=C(C=CC(S(=O)(N3CCC(CC3)C)=O)=C2)O1)NCC4=CC=C(C=C4)F

Shipping

Room temperature in continental US; may vary elsewhere.

Storage

4°C, protect from light

*In solvent : -80°C, 6 months; -20°C, 1 month (protect from light)

Solvent & Solubility

In Vitro:

DMSO : ≥ 100 mg/mL (224.96 mM; Hygroscopic DMSO has a significant impact on the solubility of product, please use newly opened DMSO)

*"≥" means soluble, but saturation unknown.

Preparing
Stock Solutions

Concentration Solvent Mass	1 mg	5 mg	10 mg

1 mM	2.2496 mL	11.2481 mL	22.4962 mL
5 mM	0.4499 mL	2.2496 mL	4.4992 mL
10 mM	0.2250 mL	1.1248 mL	2.2496 mL

View the Complete Stock Solution Preparation Table

* Please refer to the solubility information to select the appropriate solvent. Once prepared, please aliquot and store the solution to prevent product inactivation from repeated freeze-thaw cycles.
Storage method and period of stock solution: -80°C, 6 months; -20°C, 1 month (protect from light). When stored at -80°C, please use it within 6 months. When stored at -20°C, please use it within 1 month.

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Mass (g) = Concentration (mol/L) × Volume (L) × Molecular Weight (g/mol)

Concentration _(start) × Volume _(start) = Concentration _(final) × Volume _(final)

This equation is commonly abbreviated as: C₁V₁ = C₂V₂

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Calculation results:

Working solution concentration: mg/mL

Purity & Documentation

Purity: ≥98.0%

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Data Sheet (267 KB) SDS (251 KB)

COA (249 KB) HNMR (162 KB)

Handling Instructions (2659 KB)

References

[1]. Andreas P Termin, et al. Heterocyclic derivatives for modulation of calcium channels. Patent WO2006010008A1.

Complete Stock Solution Preparation Table

Optional Solvent	Concentration Solvent Mass	1 mg	5 mg	10 mg	25 mg

DMSO	1 mM	2.2496 mL	11.2481 mL	22.4962 mL	56.2404 mL
	5 mM	0.4499 mL	2.2496 mL	4.4992 mL	11.2481 mL
	10 mM	0.2250 mL	1.1248 mL	2.2496 mL	5.6240 mL
	15 mM	0.1500 mL	0.7499 mL	1.4997 mL	3.7494 mL
	20 mM	0.1125 mL	0.5624 mL	1.1248 mL	2.8120 mL
	25 mM	0.0900 mL	0.4499 mL	0.8998 mL	2.2496 mL
	30 mM	0.0750 mL	0.3749 mL	0.7499 mL	1.8747 mL
	40 mM	0.0562 mL	0.2812 mL	0.5624 mL	1.4060 mL
	50 mM	0.0450 mL	0.2250 mL	0.4499 mL	1.1248 mL
	60 mM	0.0375 mL	0.1875 mL	0.3749 mL	0.9373 mL
	80 mM	0.0281 mL	0.1406 mL	0.2812 mL	0.7030 mL
	100 mM	0.0225 mL	0.1125 mL	0.2250 mL	0.5624 mL