2. GPCR/G Protein Neuronal Signaling Immunology/Inflammation
  3. Histamine Receptor
  4. Antazoline phosphate

Antazoline phosphate  (Synonyms: Phenazoline phosphate)

Cat. No.: HY-B1067B
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Antazoline (phosphate) is an H1 receptor antagonist that affects the activity of the central nervous system, has a potent antiarrhythmic effect.

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Antazoline phosphate Chemical Structure

Antazoline phosphate Chemical Structure

CAS No. : 154-68-7

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Antazoline phosphate Related Antibodies

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Description

Antazoline (phosphate) is an H1 receptor antagonist that affects the activity of the central nervous system, has a potent antiarrhythmic effect[1][2][3].

In Vitro

Antazoline (phosphate) shows good inhibitory effect on HBV DNA in the supernatant of HepAD38 and Huh7 cells with the value of EC50 is 2.910 μmol/L and 2.349 μmol/L, respectively[2].

MedChemExpress (MCE) has not independently confirmed the accuracy of these methods. They are for reference only.

Antazoline phosphate Related Antibodies

Cell Viability Assay[2]

Cell Line: HepAD38 cells
Concentration: 10 μmol/L
Incubation Time: 5 days
Result: Exhibited no significant cytotoxicity at a concentration of 10μmol/L and had a dose-dependent inhibition of HBV DNA in the supernatant.

RT-PCR[2]

Cell Line: Huh7 cells
Concentration: 30 μmol/L, 10 μmol/L, 3.33 μmol/L, 1.1 μmol/L, 0.370 μmol/L, and 0.123 μmol/L
Incubation Time: 4 days
Result: Had a significant inhibitory effect on HBV DNA in supernatants in a dose-dependent manner.
In Vivo

Antazoline (phosphate) (IP; 0.01 ml/g; 30min) as H1 receptor antagonists diminishes the anticonvulsant activity of carbamazepine and diphenylhydantoin[3].

MedChemExpress (MCE) has not independently confirmed the accuracy of these methods. They are for reference only.

Animal Model: Swiss mice[3]
Dosage: 0.01 mL/g
Administration: IP; 0.01 ml/g; 30min
Result: Showed some proconvulsive activity.
Molecular Weight

363.35

Formula

C17H22N3O4P
CAS No.
SMILES

O=P(O)(O)O.C1(CN(C2=CC=CC=C2)CC3=CC=CC=C3)=NCCN1
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Room temperature in continental US; may vary elsewhere.
Storage

Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
References
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Antazoline phosphate Related Classifications

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The molarity calculator equation

Mass (g) = Concentration (mol/L) × Volume (L) × Molecular Weight (g/mol)

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The dilution calculator equation

Concentration (start) × Volume (start) = Concentration (final) × Volume (final)

This equation is commonly abbreviated as: C1V1 = C2V2

Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
× = ×
C1   V1   C2   V2
Help & FAQs
  • Do most proteins show cross-species activity?

    Species cross-reactivity must be investigated individually for each product. Many human cytokines will produce a nice response in mouse cell lines, and many mouse proteins will show activity on human cells. Other proteins may have a lower specific activity when used in the opposite species.

Keywords:

Antazoline154-68-7PhenazolineHistamine ReceptorH1 receptor antagonistnervous systemInhibitorinhibitorinhibit

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