2. Signaling Pathways
  3. Metabolic Enzyme/Protease
  4. PCSK9
  5. PCSK9 Degrader

PCSK9 Degrader

PCSK9 Degraders (2):

Cat. No. Product Name Effect Purity
  • HY-130245
    PCSK9 degrader 1
    		Degrader 98.26%
    PCSK9 degrader 1 (Compound 16) is a small molecule ligand for proprotein convertase substilisin-like/kexin type 9 (PCSK9) and shows high affinity to PCSK9 with a Ki of 107 nM. PCSK9 degrader 1 can involve in a protein-protein interaction with the low-density lipoprotein (LDL) receptor.
  • HY-130245A
    (R,R)-PCSK9 degrader 1
    		Degrader
    (R,R)-PCSK9 degrader 1 is the isomer of PCSK9 degrader 1 (HY-130245). PCSK9 degrader 1 (Compound 16) is a small molecule ligand for proprotein convertase substilisin-like/kexin type 9 (PCSK9) and shows high affinity to PCSK9 with a Ki of 107 nM. PCSK9 degrader 1 can involve in a protein-protein interaction with the low-density lipoprotein (LDL) receptor.