1. Others GPCR/G Protein Autophagy
  2. Isotope-Labeled Compounds Angiotensin Receptor Autophagy
  3. Telmisartan-13C,d3

Telmisartan-13C,d3  (Synonyms: BIBR 277-13C,d3)

Cat. No.: HY-13955S2
Handling Instructions

Telmisartan-13C,d3 is the 13C- and deuterium labeled Telmisartan. Telmisartan is a potent, long lasting antagonist of angiotensin II type 1 receptor (AT1), selectively inhibiting the binding of 125I-AngII to AT1 receptors with IC50 of 9.2 nM.

For research use only. We do not sell to patients.

Telmisartan-<sup>13</sup>C,d<sub>3</sub> Chemical Structure

Telmisartan-13C,d3 Chemical Structure

CAS No. : 1261396-33-1

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Description

Telmisartan-13C,d3 is the 13C- and deuterium labeled Telmisartan. Telmisartan is a potent, long lasting antagonist of angiotensin II type 1 receptor (AT1), selectively inhibiting the binding of 125I-AngII to AT1 receptors with IC50 of 9.2 nM.

In Vitro

Stable heavy isotopes of hydrogen, carbon, and other elements have been incorporated into drug molecules, largely as tracers for quantitation during the drug development process. Deuteration has gained attention because of its potential to affect the pharmacokinetic and metabolic profiles of drugs[55].

MedChemExpress (MCE) has not independently confirmed the accuracy of these methods. They are for reference only.

Molecular Weight

518.63

Formula

C3213CH27D3N4O2

CAS No.
Unlabeled CAS

144701-48-4

SMILES

CCCC(N(C1=CC(C2=NC3=CC=CC=C3N2[13C]([2H])([2H])[2H])=C4)CC5=CC=C(C6=C(C=CC=C6)C(O)=O)C=C5)=NC1=C4C

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Room temperature in continental US; may vary elsewhere.

Storage

Please store the product under the recommended conditions in the Certificate of Analysis.

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Telmisartan-13C,d3
Cat. No.:
HY-13955S2
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